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Opioid Analgesic Info Tables

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Information on dosage, duration, scheduling.


From: Marco Manzo
Newsgroups: alt.drugs
Subject: FAQ list-Opioid Analgesics
Date: 29 May 1994 19:16:02 GMT
Message-ID: <2sapli$nca@netnews.upenn.edu>

CATEGORY I. STRONG AGONISTS-- SEVERE PAIN
GENERIC NAMETRADE NAMEDOSAGEDURATION OF ACTIONCONTROLLED SUBSTANCE CATEGORY
HYDROMORPHONEDILAUDID2-4 mg. every 4-6 hrs4-5 hoursSchedule II Narcotic
avail in: 1,2,3,4,10 mg.tabs Parenteral (injection) 1,2,3,4 mg./mL ampules
LEVORPHANOLLEVO-DROMORAN2-3 mg. every 6-8 hrs.4-5 hoursSchedule II Narcotic
dosages: 2 mg. tabs; injection: 2 mg./mL
MEPERIDINEDEMEROL50-150 mg. every 3-4 hrs2-4 hoursSchedule II Narcotic
dosages: 50,100 mg. tabs; injection: 25,50,75,100 mg. vials
METHADONEDOLOPHINE40 mg. every 24 hrs4-6 hoursSchedule II Narcotic
dosages: 5,10,40 mg. tabs; injection: 10 mg./mL 2.5-10 mg.injection every 3-4 hrs
MORPHINESULFATE10-30 mg. every 4 hrs4-5 hoursSchedule II Narcotic
dosages: 10,15,30 mg., tabs injection: 2,4,5,8,10,15 mg/mL, 30 mg. controlled release tablets 8-12 hrs.
OXYMORPHONENUMORPHON5 mg. suppository every 4-6 hours3-4 hoursSchedule II Narcotic
dosages: 5 mg. suppos., 1, 1.5 mg/mL injection, 1-1.5 mg. injection every 4-6 hours

STRONG AGONISTS FOR INJECTION ONLY:
GENERIC NAMETRADE NAMEDOSAGEDURATION OF ACTIONCONTROLLED SUBSTANCE CATEGORY
FENTANYLSUBLIMAZE0.05-0.1 mg.1-1.5 hoursSchedule II Narcotic
dosages: 0.05 mL for injectionrepeat in 2 hours if needed
SUFENTANILSUFENTA1-30 micrograms/kg. as needed for anesthesiaSchedule II Narcotic
dosages: 50 micrograms per mL in 1,2,5 mL ampules
ALFENTANILALFENTA0.5-3 micrograms/kg./minuteSchedule II Narcotic
dosage: 500 micrograms/mL ampules for injectionIV infusion in balanced anesthesia

CATEGORY II, MILD TO MODERATE AGONISTS, MODERATE TO SEVERE PAIN
GENERIC NAMETRADE NAMEDOSAGEDURATION OF ACTIONCONTROLLED SUBSTANCE CATEGORY
CODEINESULFATE,PHOSPHATE15-60 mg. every 4-6 hours3-4 hoursSchedule II Narcotic
dosage 15,30,60 mg. tablets 30,60 mg./mL for injection(when combined with acetaminophen or asprin it is a Schedule III Narcotic)
OXYCODONEPERCODAN (with asprin)5 mg.3-4 hoursSchedule II Narcotic
dosage 5 mg. oxycodone per tabletPERCOCET (with tylenol)every 6 hours
HYDROCODONEVICODIN,LORTAB5-7 mg.3-4 hoursSchedule III Narcotic
BITARTRATELORCET,HYDROCET5-7 mg.4-6 hours
dosages: either 2.5, 5, or 7 mg. hydrocodone with either asprin or tylenol

CATEGORY III, WEAK AGONISTS, MILD TO MODERATE PAIN
GENERIC NAMETRADE NAMEDOSAGEDURATION OF ACTIONCONTROLLED SUBSTANCE CATEGORY
PROPOXYPHENEDARVON50-100 mg. every 4 hrs4-5 hoursSchedule IV Narcotic
NAPSYLATEDARVOCET N-50
DARVOCET N-100

CATEGORY IV, MIXED AGONISTS/ANTAGONISTS, MODERATE TO SEVERE PAIN
GENERIC NAMETRADE NAMEDOSAGEDURATION OF ACTIONCONTROLLED SUBSTANCE CATEGORY
PENTAZOCINETALWIN-NX50-100 mg.3 hoursSchedule IV Narcotic
dosage 50 mg. tablets, 30 mg./mL in 1 and 2 mL ampules for injectionevery 3-4 hours 30 mg. injection (Pentazocine is mixed with Naxolone [an opiate antagonist] to prevent crushing of tabs. for iv injection)

OTHER MIXED AGONIST-ANTAGONISTS:
GENERIC NAMETRADE NAMEDOSAGEDURATION OF ACTIONCONTROLLED SUBSTANCE CATEGORY
BUPRENORPHINEBUPRENEX0.3 mg./ml ampules for injectionSchedule V
BUTORPHANOLSTADOL1-2 mg./ml for injectionNot a controlled substance because of the strong antagonist efficacy
NALBUPHINENUBAIN10-20 mg./ml for injectionNot a controlled substance because of the strong antagonist efficacy

Created 10/12/2000 18:45:19
Modified 10/12/2000 18:51:58
Leda version 1.4.3