|
The New Lycaeum
What's New
Announcements
Disclaimer
Leda
About Leda
Chemicals
Taxonomy
Preparations
Categories
Links
Lycaeum
Homepage
Forums
Chat
Hosted Sites
Books
Contact
About
|
Information on dosage, duration, scheduling.
From: Marco Manzo
Newsgroups: alt.drugs
Subject: FAQ list-Opioid Analgesics
Date: 29 May 1994 19:16:02 GMT
Message-ID: <2sapli$nca@netnews.upenn.edu>
| CATEGORY I. STRONG AGONISTS-- SEVERE PAIN |
| GENERIC NAME | TRADE NAME | DOSAGE | DURATION OF ACTION | CONTROLLED SUBSTANCE CATEGORY |
| HYDROMORPHONE | DILAUDID | 2-4 mg. every 4-6 hrs | 4-5 hours | Schedule II Narcotic |
| avail in: 1,2,3,4,10 mg.tabs Parenteral (injection) 1,2,3,4 mg./mL ampules |
| LEVORPHANOL | LEVO-DROMORAN | 2-3 mg. every 6-8 hrs. | 4-5 hours | Schedule II Narcotic |
| dosages: 2 mg. tabs; injection: 2 mg./mL |
| MEPERIDINE | DEMEROL | 50-150 mg. every 3-4 hrs | 2-4 hours | Schedule II Narcotic |
| dosages: 50,100 mg. tabs; injection: 25,50,75,100 mg. vials |
| METHADONE | DOLOPHINE | 40 mg. every 24 hrs | 4-6 hours | Schedule II Narcotic |
| dosages: 5,10,40 mg. tabs; injection: 10 mg./mL 2.5-10 mg.injection every 3-4 hrs |
| MORPHINE | SULFATE | 10-30 mg. every 4 hrs | 4-5 hours | Schedule II Narcotic |
| dosages: 10,15,30 mg., tabs injection: 2,4,5,8,10,15 mg/mL, 30 mg. controlled release tablets 8-12 hrs. |
| OXYMORPHONE | NUMORPHON | 5 mg. suppository every 4-6 hours | 3-4 hours | Schedule II Narcotic |
| dosages: 5 mg. suppos., 1, 1.5 mg/mL injection, 1-1.5 mg. injection every 4-6 hours |
| STRONG AGONISTS FOR INJECTION ONLY: |
| GENERIC NAME | TRADE NAME | DOSAGE | DURATION OF ACTION | CONTROLLED SUBSTANCE CATEGORY |
| FENTANYL | SUBLIMAZE | 0.05-0.1 mg. | 1-1.5 hours | Schedule II Narcotic |
| dosages: 0.05 mL for injection | repeat in 2 hours if needed |
| SUFENTANIL | SUFENTA | 1-30 micrograms/kg. as needed for anesthesia | Schedule II Narcotic |
| dosages: 50 micrograms per mL in 1,2,5 mL ampules |
| ALFENTANIL | ALFENTA | 0.5-3 micrograms/kg./minute | Schedule II Narcotic |
| dosage: 500 micrograms/mL ampules for injection | IV infusion in balanced anesthesia |
| CATEGORY II, MILD TO MODERATE AGONISTS, MODERATE TO SEVERE PAIN |
| GENERIC NAME | TRADE NAME | DOSAGE | DURATION OF ACTION | CONTROLLED SUBSTANCE CATEGORY |
| CODEINE | SULFATE,PHOSPHATE | 15-60 mg. every 4-6 hours | 3-4 hours | Schedule II Narcotic |
| dosage 15,30,60 mg. tablets 30,60 mg./mL for injection | (when combined with acetaminophen or asprin it is a Schedule III Narcotic) |
| OXYCODONE | PERCODAN (with asprin) | 5 mg. | 3-4 hours | Schedule II Narcotic |
| dosage 5 mg. oxycodone per tablet | PERCOCET (with tylenol) | every 6 hours |
| HYDROCODONE | VICODIN,LORTAB | 5-7 mg. | 3-4 hours | Schedule III Narcotic |
| BITARTRATE | LORCET,HYDROCET | 5-7 mg. | 4-6 hours |
| dosages: either 2.5, 5, or 7 mg. hydrocodone with either asprin or tylenol |
| CATEGORY III, WEAK AGONISTS, MILD TO MODERATE PAIN |
| GENERIC NAME | TRADE NAME | DOSAGE | DURATION OF ACTION | CONTROLLED SUBSTANCE CATEGORY |
| PROPOXYPHENE | DARVON | 50-100 mg. every 4 hrs | 4-5 hours | Schedule IV Narcotic |
| NAPSYLATE | DARVOCET N-50 DARVOCET N-100 |
| CATEGORY IV, MIXED AGONISTS/ANTAGONISTS, MODERATE TO SEVERE PAIN
|
| GENERIC NAME | TRADE NAME | DOSAGE | DURATION OF ACTION | CONTROLLED SUBSTANCE CATEGORY |
| PENTAZOCINE | TALWIN-NX | 50-100 mg. | 3 hours | Schedule IV Narcotic |
dosage 50 mg. tablets, 30 mg./mL in 1 and 2 mL ampules for injection | every 3-4 hours 30 mg. injection (Pentazocine is mixed with Naxolone [an opiate antagonist] to prevent crushing of tabs. for iv injection) |
| OTHER MIXED AGONIST-ANTAGONISTS: |
| GENERIC NAME | TRADE NAME | DOSAGE | DURATION OF ACTION | CONTROLLED SUBSTANCE CATEGORY |
| BUPRENORPHINE | BUPRENEX | 0.3 mg./ml ampules for injection | Schedule V |
BUTORPHANOL | STADOL | 1-2 mg./ml for injection | Not a controlled substance because of the strong antagonist efficacy |
| NALBUPHINE | NUBAIN | 10-20 mg./ml for injection | Not a controlled substance because of the strong antagonist efficacy |
Created 10/12/2000 18:45:19 Modified 10/12/2000 18:51:58 | Leda version 1.4.3 |
|